G-PROTEIN-COUPLED-RECEPTOR
- 2P-125 Poster: October 20 (Thu) 17:00 Room Poster (Hall No.1 1F/2F, Hall No.2 1F, Kobe International Exhibition Hall)
Immunosuppressive reagent FTY720 inhibits cell migration through S1P1 desensitization-independent pathways: Takayuki Kohno, Yasuyuki Igarashi Keywords: G-PROTEIN-COUPLED-RECEPTOR; DESENSITIZATION; CELL-MOTILITY
- 2P-127(WS27-9) Poster: October 20 (Thu) 17:00 Room Poster (Hall No.1 1F/2F, Hall No.2 1F, Kobe International Exhibition Hall) / Workshop: October 20 (Thu) 10:53 Room U (Hall No.2 3F B, Kobe International Exhibition Hall)
Extracellular Acidic pH induced SRE-driven transcription and decreased EGF-induced ERK1/2 activation in GPR4-overexpressing RH 7777 cells.: Masayuki Tobo, Hideaki Tomura, Fumikazu Okajima Keywords: G-PROTEIN-COUPLED-RECEPTOR; PH-EFFECT; VASCULAR-SMOOTH-MUSCLE-CELL
- 2P-128(WS27-10) Poster: October 20 (Thu) 17:00 Room Poster (Hall No.1 1F/2F, Hall No.2 1F, Kobe International Exhibition Hall) / Workshop: October 20 (Thu) 11:04 Room U (Hall No.2 3F B, Kobe International Exhibition Hall)
Identification of human G2A as a receptor for oxidized free fatty acids: Hideru Obinata, Tomoyasu Hattori, Shinji Nakane, Kazuaki Tatei, Takashi Izumi Keywords: G-PROTEIN-COUPLED-RECEPTOR; LIPID-MEDIATOR; ORPHAN-RECEPTOR
- 2P-129(WS27-11) Poster: October 20 (Thu) 17:00 Room Poster (Hall No.1 1F/2F, Hall No.2 1F, Kobe International Exhibition Hall) / Workshop: October 20 (Thu) 11:15 Room U (Hall No.2 3F B, Kobe International Exhibition Hall)
TG1019/OXE, a Gαi/o-protein-coupled receptor, mediates cell migration induced by 5-oxo-eicosatetraenoic acid: Takeshi Hosoi, Emiko Sugikawa, Aiko Chikada, Yutaka Koguchi, Tetsuo Ohnuki Keywords: LIPID-MEDIATOR; CHEMOTAXIS; G-PROTEIN-COUPLED-RECEPTOR
- 2P-130 Poster: October 20 (Thu) 17:00 Room Poster (Hall No.1 1F/2F, Hall No.2 1F, Kobe International Exhibition Hall)
Role of helix 8 of Leukotriene B4 receptor: Toshiaki Okuno, Takehiko Yokomizo, Tetsuya Hori, Masashi Miyano, Takao Shimizu Keywords: G-PROTEIN-COUPLED-RECEPTOR; LEUKOTRIENE; G-PROTEIN
- 2P-570 Poster: October 20 (Thu) 17:00 Room Poster (Hall No.1 1F/2F, Hall No.2 1F, Kobe International Exhibition Hall)
Key amino acid residues on the cytoplasmic surface responsible for the formation of the active state of metabotropic glutamate receptor: Takahiro Yamashita, Akihisa Terakita, Yoshinori Shichida Keywords: G-PROTEIN-COUPLED-RECEPTOR; GLUTAMATE-RECEPTOR; G-PROTEIN
- 2P-573 Poster: October 20 (Thu) 17:00 Room Poster (Hall No.1 1F/2F, Hall No.2 1F, Kobe International Exhibition Hall)
Identification of the Cysteine Residues in the Ligand Binding Site by Affinity Labeling using the Mutant δ Opioid Receptors: Kaname Isozaki, Jun-ichi Funama, Sayaka Koikawa, Hidehiko Fukahori, Takeru Nose, Tommaso Costa, Yasuyuki Shimohigashi Keywords: AFFINITY-LABELING; G-PROTEIN-COUPLED-RECEPTOR; RECEPTOR-BINDING
- 2P-587 Poster: October 20 (Thu) 17:00 Room Poster (Hall No.1 1F/2F, Hall No.2 1F, Kobe International Exhibition Hall)
N-terminal acyl-alkyl group of Ac-RYYRIK-NH2 as a structural determinant for nociceptin antagonism: Jinglan Li, Kaname Isozaki, Michiaki Kawano, Takeru Nose, Tommaso Costa, Yasuyuki Shimohigashi Keywords: ANTAGONIST; G-PROTEIN-COUPLED-RECEPTOR; RECEPTOR-BINDING
- 2P-588 Poster: October 20 (Thu) 17:00 Room Poster (Hall No.1 1F/2F, Hall No.2 1F, Kobe International Exhibition Hall)
Molecular cloning and characterization of chicken neuromedin B recepotr: Masayuki Shibayama, Kazuhiko Inoue, Hideki Sugawara, Hiroki Saito, Shin-ichi Iwata, Takao Shimizu, Atsuro Miyata Keywords: G-PROTEIN-COUPLED-RECEPTOR; NEUROMEDIN; NEUROPEPTIDE
- 2P-590 Poster: October 20 (Thu) 17:00 Room Poster (Hall No.1 1F/2F, Hall No.2 1F, Kobe International Exhibition Hall)
Hetero-oligomer formation between A1 adenosine receptor and P2Y2 receptor: Tokiko Suzuki, Kazunori Namba, Hirofumi Tsuga, Hiroyasu Nakata Keywords: ADENOSINE; G-PROTEIN-COUPLED-RECEPTOR; MEMBRANE-PROTEIN-ASSEMBLY
- 2P-591 Poster: October 20 (Thu) 17:00 Room Poster (Hall No.1 1F/2F, Hall No.2 1F, Kobe International Exhibition Hall)
The cell surface localization of thromboxane A2 receptor is regulated by proteasome: Masako Sasaki, Jun Sukegawa, Katsutoshi Miyosawa, Teruyuki Yanagisawa, Satoko Ohkubo, Norimichi Nakahata Keywords: THROMBOXANE; PROTEASOME; G-PROTEIN-COUPLED-RECEPTOR
- 2P-598 Poster: October 20 (Thu) 17:00 Room Poster (Hall No.1 1F/2F, Hall No.2 1F, Kobe International Exhibition Hall)
Expression and purification of the receptor for pituitary adenylate cyclase-activating polypeptide: Youhei Kuramochi, Hiroshi Suzuki, Tomoko Doi, Yoshinori Fujiyoshi Keywords: BACULOVIRUS; G-PROTEIN-COUPLED-RECEPTOR; PITUITARY-ADENYLATE-CYCLASE-ACTIVATING-POLYPEPTIDE
- 2P-599(WS49-5) Poster: October 20 (Thu) 17:00 Room Poster (Hall No.1 1F/2F, Hall No.2 1F, Kobe International Exhibition Hall) / Workshop: October 21 (Fri) 10:13 Room R (International Conference Room 301, International Conference Center Kobe)
Direct interaction between purinergic receptors present in platelet membranes: Koshi Oyanagi, Toshio Kamiya, Hiroyasu Nakata Keywords: G-PROTEIN-COUPLED-RECEPTOR; PLATELET; OLIGOMERIZATION
- 2P-609(WS49-10) Poster: October 20 (Thu) 17:00 Room Poster (Hall No.1 1F/2F, Hall No.2 1F, Kobe International Exhibition Hall) / Workshop: October 21 (Fri) 11:13 Room R (International Conference Room 301, International Conference Center Kobe)
Differential activation of G proteins by β2-adrenergic receptor selective agonists: Masashi Fukutomi, Kyoji Urayama, Ryuji Inoue, Motohiro Nishida, Hitoshi Kurose Keywords: ADRENERGIC-RECEPTOR; G-PROTEIN-COUPLED-RECEPTOR; G-PROTEIN
- 2P-610 Poster: October 20 (Thu) 17:00 Room Poster (Hall No.1 1F/2F, Hall No.2 1F, Kobe International Exhibition Hall)
cDNA Cloning of GPCR receptor of FMRFamide-related Peptides from the Housefly Musca domestica: Ayami Matsushima, Yukie Koretsune, Taichi Yoshida, Atsushi Kaneki, Kaname Isozaki, Miki Shimohigashi, Yasuyuki Shimohigashi Keywords: CDNA-CLONING; G-PROTEIN-COUPLED-RECEPTOR; INOSITOL-PHOSPHOLIPID
- 2P-612(WS63-2) Poster: October 20 (Thu) 17:00 Room Poster (Hall No.1 1F/2F, Hall No.2 1F, Kobe International Exhibition Hall) / Workshop: October 21 (Fri) 14:42 Room R (International Conference Room 301, International Conference Center Kobe)
Cellular Responses Elicited by Acidic Environments Through T Cell Death-Associated Gene 8 (TDAG8): Yasuyuki Kihara, Satoshi Ishii, Takao Shimizu Keywords: G-PROTEIN-COUPLED-RECEPTOR; ACID-SENSITIVE; CYCLIC-AMP
- 2P-615(WS63-4) Poster: October 20 (Thu) 17:00 Room Poster (Hall No.1 1F/2F, Hall No.2 1F, Kobe International Exhibition Hall) / Workshop: October 21 (Fri) 15:06 Room R (International Conference Room 301, International Conference Center Kobe)
Dynamin-dependent internalization of muscarinic acetylcholine receptor M4 subtype: Kanoko Morisawa, Yuichi Hashimoto, Hiroyuki Saito, Eri Jojima, Norihiro Yoshida, Tatuya Haga Keywords: G-PROTEIN-COUPLED-RECEPTOR; DYNAMIN; ACETYLCHOLINE
- 2P-616 Poster: October 20 (Thu) 17:00 Room Poster (Hall No.1 1F/2F, Hall No.2 1F, Kobe International Exhibition Hall)
Functions of clathrin box in G protein-coupled receptor kinase 2 (GRK2): Supachoke Mangmool, Motohiro Nishida, Hiroyuki Kobayashi, Tatsuya Haga, Hitoshi Kurose Keywords: G-PROTEIN-COUPLED-RECEPTOR; CLATHRIN-VESICLE; ADRENERGIC-RECEPTOR
- 3P-203(WS13-10) Poster: October 21 (Fri) 17:00 Room Poster (Hall No.1 1F/2F, Hall No.2 1F, Kobe International Exhibition Hall) / Workshop: October 19 (Wed) 18:28 Room U (Hall No.2 3F B, Kobe International Exhibition Hall)
Extracellular Acidic pH Induced Prostacyclin Production and cAMP Accumulation Through OGR1 in Human Aortic Smooth Muscle Cells: Hideaki Tomura, Ju-Qiang Wang, Mayumi Komachi, Alatangaole Damirin, Chihiro Mogi, Masayuki Tobo, Koichi Sato, Fumikazu Okajima Keywords: G-PROTEIN-COUPLED-RECEPTOR; PH-EFFECT; VASCULAR-SMOOTH-MUSCLE-CELL
- 3P-451(WS59-2) Poster: October 21 (Fri) 17:00 Room Poster (Hall No.1 1F/2F, Hall No.2 1F, Kobe International Exhibition Hall) / Workshop: October 21 (Fri) 14:42 Room K (501, International Conference Center Kobe)
Differential Regulation of Phosphorylation of the cAMP Response Element Binding Protein Following Activation of EP2 and EP4 Prostanoid Receptors by Prostaglandin E2: Hiromichi Fujino, Sambhitab Salvi, John W. Regan, Toshihiko Murayama Keywords: PROSTAGLANDIN; CREB; G-PROTEIN-COUPLED-RECEPTOR
- 3P-452 Poster: October 21 (Fri) 17:00 Room Poster (Hall No.1 1F/2F, Hall No.2 1F, Kobe International Exhibition Hall)
Analysis of the interaction between RGS8 and M1 acetylcholine receptor: Masayuki Itoh, Osamu Saitoh Keywords: REGULATOR-OF-G-PROTEIN-SIGNALING; G-PROTEIN; G-PROTEIN-COUPLED-RECEPTOR
- 3P-733 Poster: October 21 (Fri) 17:00 Room Poster (Hall No.1 1F/2F, Hall No.2 1F, Kobe International Exhibition Hall)
Structure of the third intracellular loop of the muscarinic acetylcholine receptor M2 subtype: Susumu Ichiyama, Yoshiaki Oka, Kazuko Haga, Shuichi Kojima, Yukihiro Tateishi, Masahiro Shirakawa, Tatsuya Haga Keywords: ACETYLCHOLINE-RECEPTOR; G-PROTEIN-COUPLED-RECEPTOR; STRUCTURE